Bupivacaine

Local Anesthetics

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Calculated Induction Dose
--mg

Mechanism of Action

Highly potent, long-acting amide LA. Carries a high risk of severe cardiotoxicity (refractory arrhythmias) if injected intravascularly due to slow dissociation from cardiac sodium channels.

Dosage Guidelines

TypeRouteRate / Dose
Dosage/GuidelineSystemicMax dose: 3 mg/kg.

Clinical Pearls

1

Highly potent, highly lipid-soluble with slow onset and long duration. Lipid emulsion (Intralipid 20%) is a first-line rescue treatment for cardiovascular toxicity.

Population Considerations